c-Fms抑制劑|c-Fms
c-FMS(CSF1R,CSF-1R)位于細(xì)胞質(zhì)膜上。c-FMS是配體集落刺激因子-1(CSF1)的受體。c-FMS是一種完整的跨膜糖蛋白,具有配體誘導(dǎo)的酪氨酸特異性蛋白激酶活性,從而觸發(fā)信號(hào)級(jí)聯(lián),最終影響CSF1應(yīng)答基因的轉(zhuǎn)錄。c-FMS酪氨酸磷酸化在CSF1結(jié)合時(shí)被誘導(dǎo),導(dǎo)致Ras/Erk和I-A類磷脂酰肌醇3激酶信號(hào)通路的激活,進(jìn)而激活信號(hào)轉(zhuǎn)導(dǎo)和轉(zhuǎn)錄激活(STATs)通路,特別是STAT1、STAT3和STAT5。CSF1激活c-FMS可促進(jìn)生長(zhǎng)、增殖和分化。
c-Fms抑制劑
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